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Brexpiprazole, MedChemExpress

Product Code. 16406946
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Product Code. 16406946

Brand: Medchem Express HY15780

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Description

MedChemExpress Brexpiprazole (OPC-34712), an atypical orally active antipsychotic drug, is a partial agonist of human 5-HT1A and dopamine D2L receptor with Kis of 0.12 nM and 0.3 nM, respectively. Brexpiprazole is also a 5-HT2A receptor antagonist with a Ki of 0.47 nM. Brexpiprazole also shows potent antagonist activity at human noradrenergic α1B (Ki=0.17 nM) and α2C receptors (Ki=0.59 nM).

Brexpiprazole (OPC-34712), an atypical orally active antipsychotic drug, is a partial agonist of human 5-HT1A and dopamine D2L receptor with Kis of 0.12 nM and 0.3 nM, respectively. Brexpiprazole is also a 5-HT2A receptor antagonist with a Ki of 0.47 nM. Brexpiprazole also shows potent antagonist activity at human noradrenergic α1B (Ki=0.17 nM) and α2C receptors (Ki=0.59 nM).

Specifications

Materiale o nome chimico Brexpiprazole
CAS 913611-97-9
Colore White
Note sul grado di purezza Research
Formula molecolare C25H27N3O2S
Quantità 100 mg
Sinonimo OPC-34712
Informazioni di solubilità DMSO : 25 mg/mL (57.66 mM; ultrasonic and warming and heat to 80°C)
SMILES O=C1NC2=C(C=CC(OCCCCN3CCN(C4=C(C=CS5)C5=CC=C4)CC3)=C2)C=C1
Molecular Weight (g/mol) 433.57
Peso formulazione 433.57
Percent Purity 98.25%
Grado Research
Forma fisica Powder
Da utilizzare con (applicazione) Neuroscience-Neuromodulation
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Research purposes only

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